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Example Input Mode:
Partner Data
CBIS
Matrix
Example Data Type:
Secondary Screen (Kd)
Primary Screen(% control or competition)
If the input file contains Primary and Secondary Data, use:
Primary
Secondary
Assay Data File:
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Bromodomain
Kd
Primary
To highlight spots, select a compound(s), click 'fill' and select entries.
Create Images for:
PHA-665752
Highlight These Spots (
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):
PHA-665752|AAK1|320
PHA-665752|ABL1-nonphosphorylated|2600
PHA-665752|ABL2|6900
PHA-665752|ALK|2700
PHA-665752|AMPK-alpha1|310
PHA-665752|AMPK-alpha2|770
PHA-665752|ARK5|620
PHA-665752|AURKB|2000
PHA-665752|AURKC|300
PHA-665752|AXL|110
PHA-665752|BIKE|47
PHA-665752|BLK|1900
PHA-665752|BMPR2|6200
PHA-665752|CAMK1|2100
PHA-665752|CAMK1D|1500
PHA-665752|CAMK2A|3400
PHA-665752|CAMK2D|2900
PHA-665752|CAMK2G|2000
PHA-665752|CAMKK1|64
PHA-665752|CAMKK2|73
PHA-665752|CASK|1700
PHA-665752|CDK4-cyclinD1|2500
PHA-665752|CDK7|130
PHA-665752|CDK9|1800
PHA-665752|CDKL2|2400
PHA-665752|CLK1|730
PHA-665752|CLK2|410
PHA-665752|CLK3|3600
PHA-665752|CSF1R|700
PHA-665752|CSNK1D|4200
PHA-665752|CSNK1E|860
PHA-665752|CSNK2A2|5600
PHA-665752|DCAMKL1|1400
PHA-665752|DCAMKL2|990
PHA-665752|DCAMKL3|4500
PHA-665752|DDR1|70
PHA-665752|DDR2|7600
PHA-665752|DLK|670
PHA-665752|DRAK1|4000
PHA-665752|DRAK2|3500
PHA-665752|EPHA8|3900
PHA-665752|EPHB6|2900
PHA-665752|ERK5|1700
PHA-665752|FAK|1900
PHA-665752|FGFR2|5200
PHA-665752|FGFR3|5200
PHA-665752|FGR|1900
PHA-665752|FLT3|250
PHA-665752|FLT4|1400
PHA-665752|GAK|1300
PHA-665752|GCN2(Kin.Dom.2,S808G)|3400
PHA-665752|GRK1|1100
PHA-665752|GRK4|420
PHA-665752|GRK7|61
PHA-665752|HIPK1|93
PHA-665752|HIPK2|120
PHA-665752|HIPK3|63
PHA-665752|HIPK4|1300
PHA-665752|HPK1|150
PHA-665752|HUNK|1400
PHA-665752|ICK|400
PHA-665752|IKK-epsilon|700
PHA-665752|INSR|2300
PHA-665752|INSRR|3500
PHA-665752|IRAK1|1600
PHA-665752|IRAK3|610
PHA-665752|IRAK4|2500
PHA-665752|JAK1(JH2domain-pseudokinase)|2700
PHA-665752|JAK2(JH1domain-catalytic)|430
PHA-665752|JAK3(JH1domain-catalytic)|470
PHA-665752|KIT|3200
PHA-665752|LCK|320
PHA-665752|LKB1|2600
PHA-665752|LOK|290
PHA-665752|LZK|3200
PHA-665752|MAK|890
PHA-665752|MAP3K2|5200
PHA-665752|MAP3K3|5900
PHA-665752|MAP3K4|1800
PHA-665752|MAP4K2|3600
PHA-665752|MAP4K3|490
PHA-665752|MAP4K4|280
PHA-665752|MAP4K5|79
PHA-665752|MARK2|3600
PHA-665752|MEK1|1100
PHA-665752|MEK2|980
PHA-665752|MEK5|1400
PHA-665752|MERTK|1300
PHA-665752|MET|0.27
PHA-665752|MINK|250
PHA-665752|MST1R|2000
PHA-665752|MST2|1900
PHA-665752|MST4|3800
PHA-665752|MYLK|7900
PHA-665752|MYLK2|960
PHA-665752|NEK2|600
PHA-665752|NIM1|8700
PHA-665752|PAK1|2900
PHA-665752|PAK3|1100
PHA-665752|PAK7|2600
PHA-665752|PCTK1|1100
PHA-665752|PCTK2|880
PHA-665752|PCTK3|1500
PHA-665752|PDGFRA|2000
PHA-665752|PDGFRB|1900
PHA-665752|PFTAIRE2|510
PHA-665752|PFTK1|1300
PHA-665752|PHKG1|1900
PHA-665752|PHKG2|2400
PHA-665752|PIP5K1A|280
PHA-665752|PIP5K2B|1600
PHA-665752|PLK2|8300
PHA-665752|PLK4|410
PHA-665752|PRP4|2600
PHA-665752|PYK2|910
PHA-665752|RET|690
PHA-665752|RIOK1|470
PHA-665752|RIOK3|390
PHA-665752|RIPK1|1500
PHA-665752|ROCK2|8700
PHA-665752|ROS1|3000
PHA-665752|RPS6KA5(Kin.Dom.2-C-terminal)|1100
PHA-665752|RSK2(Kin.Dom.1-N-terminal)|9900
PHA-665752|RSK4(Kin.Dom.1-N-terminal)|6800
PHA-665752|S6K1|4100
PHA-665752|SIK2|2500
PHA-665752|SLK|350
PHA-665752|SNARK|910
PHA-665752|SRPK1|41
PHA-665752|SRPK2|500
PHA-665752|SRPK3|1600
PHA-665752|STK16|4800
PHA-665752|STK33|840
PHA-665752|TAK1|5300
PHA-665752|TAOK1|460
PHA-665752|TAOK2|1200
PHA-665752|TAOK3|43
PHA-665752|TBK1|970
PHA-665752|TIE1|1200
PHA-665752|TIE2|6700
PHA-665752|TNIK|310
PHA-665752|TRKA|320
PHA-665752|TRKB|800
PHA-665752|TRKC|930
PHA-665752|TSSK1B|2100
PHA-665752|TYK2(JH2domain-pseudokinase)|6600
PHA-665752|TYRO3|2000
PHA-665752|ULK1|2000
PHA-665752|ULK2|1500
PHA-665752|YES|1400
PHA-665752|YSK4|78
PHA-665752|AAK1
PHA-665752|ABL1-nonphosphorylated
PHA-665752|ABL2
PHA-665752|ALK
PHA-665752|AMPK-alpha1
PHA-665752|AMPK-alpha2
PHA-665752|ARK5
PHA-665752|AURKB
PHA-665752|AURKC
PHA-665752|AXL
PHA-665752|BIKE
PHA-665752|BLK
PHA-665752|BMPR2
PHA-665752|CAMK1
PHA-665752|CAMK1D
PHA-665752|CAMK2A
PHA-665752|CAMK2D
PHA-665752|CAMK2G
PHA-665752|CAMKK1
PHA-665752|CAMKK2
PHA-665752|CASK
PHA-665752|CDK4-cyclinD1
PHA-665752|CDK7
PHA-665752|CDK9
PHA-665752|CDKL2
PHA-665752|CLK1
PHA-665752|CLK2
PHA-665752|CLK3
PHA-665752|CSF1R
PHA-665752|CSNK1D
PHA-665752|CSNK1E
PHA-665752|CSNK2A2
PHA-665752|DCAMKL1
PHA-665752|DCAMKL2
PHA-665752|DCAMKL3
PHA-665752|DDR1
PHA-665752|DDR2
PHA-665752|DLK
PHA-665752|DRAK1
PHA-665752|DRAK2
PHA-665752|EPHA8
PHA-665752|EPHB6
PHA-665752|ERK5
PHA-665752|FAK
PHA-665752|FGFR2
PHA-665752|FGFR3
PHA-665752|FGR
PHA-665752|FLT3
PHA-665752|FLT4
PHA-665752|GAK
PHA-665752|GCN2(Kin.Dom.2,S808G)
PHA-665752|GRK1
PHA-665752|GRK4
PHA-665752|GRK7
PHA-665752|HIPK1
PHA-665752|HIPK2
PHA-665752|HIPK3
PHA-665752|HIPK4
PHA-665752|HPK1
PHA-665752|HUNK
PHA-665752|ICK
PHA-665752|IKK-epsilon
PHA-665752|INSR
PHA-665752|INSRR
PHA-665752|IRAK1
PHA-665752|IRAK3
PHA-665752|IRAK4
PHA-665752|JAK1(JH2domain-pseudokinase)
PHA-665752|JAK2(JH1domain-catalytic)
PHA-665752|JAK3(JH1domain-catalytic)
PHA-665752|KIT
PHA-665752|LCK
PHA-665752|LKB1
PHA-665752|LOK
PHA-665752|LZK
PHA-665752|MAK
PHA-665752|MAP3K2
PHA-665752|MAP3K3
PHA-665752|MAP3K4
PHA-665752|MAP4K2
PHA-665752|MAP4K3
PHA-665752|MAP4K4
PHA-665752|MAP4K5
PHA-665752|MARK2
PHA-665752|MEK1
PHA-665752|MEK2
PHA-665752|MEK5
PHA-665752|MERTK
PHA-665752|MET
PHA-665752|MINK
PHA-665752|MST1R
PHA-665752|MST2
PHA-665752|MST4
PHA-665752|MYLK
PHA-665752|MYLK2
PHA-665752|NEK2
PHA-665752|NIM1
PHA-665752|PAK1
PHA-665752|PAK3
PHA-665752|PAK7
PHA-665752|PCTK1
PHA-665752|PCTK2
PHA-665752|PCTK3
PHA-665752|PDGFRA
PHA-665752|PDGFRB
PHA-665752|PFTAIRE2
PHA-665752|PFTK1
PHA-665752|PHKG1
PHA-665752|PHKG2
PHA-665752|PIP5K1A
PHA-665752|PIP5K2B
PHA-665752|PLK2
PHA-665752|PLK4
PHA-665752|PRP4
PHA-665752|PYK2
PHA-665752|RET
PHA-665752|RIOK1
PHA-665752|RIOK3
PHA-665752|RIPK1
PHA-665752|ROCK2
PHA-665752|ROS1
PHA-665752|RPS6KA5(Kin.Dom.2-C-terminal)
PHA-665752|RSK2(Kin.Dom.1-N-terminal)
PHA-665752|RSK4(Kin.Dom.1-N-terminal)
PHA-665752|S6K1
PHA-665752|SIK2
PHA-665752|SLK
PHA-665752|SNARK
PHA-665752|SRPK1
PHA-665752|SRPK2
PHA-665752|SRPK3
PHA-665752|STK16
PHA-665752|STK33
PHA-665752|TAK1
PHA-665752|TAOK1
PHA-665752|TAOK2
PHA-665752|TAOK3
PHA-665752|TBK1
PHA-665752|TIE1
PHA-665752|TIE2
PHA-665752|TNIK
PHA-665752|TRKA
PHA-665752|TRKB
PHA-665752|TRKC
PHA-665752|TSSK1B
PHA-665752|TYK2(JH2domain-pseudokinase)
PHA-665752|TYRO3
PHA-665752|ULK1
PHA-665752|ULK2
PHA-665752|YES
PHA-665752|YSK4
PHA-665752|AAK1|320
PHA-665752|ABL1-nonphosphorylated|2600
PHA-665752|ABL2|6900
PHA-665752|ALK|2700
PHA-665752|AMPK-alpha1|310
PHA-665752|AMPK-alpha2|770
PHA-665752|ARK5|620
PHA-665752|AURKB|2000
PHA-665752|AURKC|300
PHA-665752|AXL|110
PHA-665752|BIKE|47
PHA-665752|BLK|1900
PHA-665752|BMPR2|6200
PHA-665752|CAMK1|2100
PHA-665752|CAMK1D|1500
PHA-665752|CAMK2A|3400
PHA-665752|CAMK2D|2900
PHA-665752|CAMK2G|2000
PHA-665752|CAMKK1|64
PHA-665752|CAMKK2|73
PHA-665752|CASK|1700
PHA-665752|CDK4-cyclinD1|2500
PHA-665752|CDK7|130
PHA-665752|CDK9|1800
PHA-665752|CDKL2|2400
PHA-665752|CLK1|730
PHA-665752|CLK2|410
PHA-665752|CLK3|3600
PHA-665752|CSF1R|700
PHA-665752|CSNK1D|4200
PHA-665752|CSNK1E|860
PHA-665752|CSNK2A2|5600
PHA-665752|DCAMKL1|1400
PHA-665752|DCAMKL2|990
PHA-665752|DCAMKL3|4500
PHA-665752|DDR1|70
PHA-665752|DDR2|7600
PHA-665752|DLK|670
PHA-665752|DRAK1|4000
PHA-665752|DRAK2|3500
PHA-665752|EPHA8|3900
PHA-665752|EPHB6|2900
PHA-665752|ERK5|1700
PHA-665752|FAK|1900
PHA-665752|FGFR2|5200
PHA-665752|FGFR3|5200
PHA-665752|FGR|1900
PHA-665752|FLT3|250
PHA-665752|FLT4|1400
PHA-665752|GAK|1300
PHA-665752|GCN2(Kin.Dom.2,S808G)|3400
PHA-665752|GRK1|1100
PHA-665752|GRK4|420
PHA-665752|GRK7|61
PHA-665752|HIPK1|93
PHA-665752|HIPK2|120
PHA-665752|HIPK3|63
PHA-665752|HIPK4|1300
PHA-665752|HPK1|150
PHA-665752|HUNK|1400
PHA-665752|ICK|400
PHA-665752|IKK-epsilon|700
PHA-665752|INSR|2300
PHA-665752|INSRR|3500
PHA-665752|IRAK1|1600
PHA-665752|IRAK3|610
PHA-665752|IRAK4|2500
PHA-665752|JAK1(JH2domain-pseudokinase)|2700
PHA-665752|JAK2(JH1domain-catalytic)|430
PHA-665752|JAK3(JH1domain-catalytic)|470
PHA-665752|KIT|3200
PHA-665752|LCK|320
PHA-665752|LKB1|2600
PHA-665752|LOK|290
PHA-665752|LZK|3200
PHA-665752|MAK|890
PHA-665752|MAP3K2|5200
PHA-665752|MAP3K3|5900
PHA-665752|MAP3K4|1800
PHA-665752|MAP4K2|3600
PHA-665752|MAP4K3|490
PHA-665752|MAP4K4|280
PHA-665752|MAP4K5|79
PHA-665752|MARK2|3600
PHA-665752|MEK1|1100
PHA-665752|MEK2|980
PHA-665752|MEK5|1400
PHA-665752|MERTK|1300
PHA-665752|MET|0.27
PHA-665752|MINK|250
PHA-665752|MST1R|2000
PHA-665752|MST2|1900
PHA-665752|MST4|3800
PHA-665752|MYLK|7900
PHA-665752|MYLK2|960
PHA-665752|NEK2|600
PHA-665752|NIM1|8700
PHA-665752|PAK1|2900
PHA-665752|PAK3|1100
PHA-665752|PAK7|2600
PHA-665752|PCTK1|1100
PHA-665752|PCTK2|880
PHA-665752|PCTK3|1500
PHA-665752|PDGFRA|2000
PHA-665752|PDGFRB|1900
PHA-665752|PFTAIRE2|510
PHA-665752|PFTK1|1300
PHA-665752|PHKG1|1900
PHA-665752|PHKG2|2400
PHA-665752|PIP5K1A|280
PHA-665752|PIP5K2B|1600
PHA-665752|PLK2|8300
PHA-665752|PLK4|410
PHA-665752|PRP4|2600
PHA-665752|PYK2|910
PHA-665752|RET|690
PHA-665752|RIOK1|470
PHA-665752|RIOK3|390
PHA-665752|RIPK1|1500
PHA-665752|ROCK2|8700
PHA-665752|ROS1|3000
PHA-665752|RPS6KA5(Kin.Dom.2-C-terminal)|1100
PHA-665752|RSK2(Kin.Dom.1-N-terminal)|9900
PHA-665752|RSK4(Kin.Dom.1-N-terminal)|6800
PHA-665752|S6K1|4100
PHA-665752|SIK2|2500
PHA-665752|SLK|350
PHA-665752|SNARK|910
PHA-665752|SRPK1|41
PHA-665752|SRPK2|500
PHA-665752|SRPK3|1600
PHA-665752|STK16|4800
PHA-665752|STK33|840
PHA-665752|TAK1|5300
PHA-665752|TAOK1|460
PHA-665752|TAOK2|1200
PHA-665752|TAOK3|43
PHA-665752|TBK1|970
PHA-665752|TIE1|1200
PHA-665752|TIE2|6700
PHA-665752|TNIK|310
PHA-665752|TRKA|320
PHA-665752|TRKB|800
PHA-665752|TRKC|930
PHA-665752|TSSK1B|2100
PHA-665752|TYK2(JH2domain-pseudokinase)|6600
PHA-665752|TYRO3|2000
PHA-665752|ULK1|2000
PHA-665752|ULK2|1500
PHA-665752|YES|1400
PHA-665752|YSK4|78
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PHA-665752
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PHA-665752
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* WildType kinase assays appear in both the main TREEspot and Mutant kinase dendrogams.
Human Kinome image created by KINOMEscan.
2 images created. To download (copy and paste) all images to your local machine click Open/Browse Image Folder.
Images Saved To:
D:\Eurofins\PROD\Applications\FrontOffice_Discovery\StudyManagement\TreeSpot\HTSTools\TreeImages\559_2rcvcbnf0oqpjling4jvpmyw\
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PHA-665752
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AAK1
ABL1-nonphosphorylated
ABL1-nonphosphorylated
ALK
ALK
AMPK-alpha1
AMPK-alpha2
ARK5
AURKB
AURKC
AXL
BIKE
BLK
CAMK1
CAMK1D
CAMK2D
CAMK2G
CAMKK1
CAMKK2
CASK
CDK4-cyclinD1
CDK7
CDK9
CDKL2
CLK1
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CSF1R
CSNK1E
DCAMKL1
DCAMKL2
DDR1
DLK
EPHB6
ERK5
FAK
FGR
FLT3
FLT3
FLT4
GAK
GRK1
GRK4
GRK7
HIPK1
HIPK2
HIPK3
HIPK4
HPK1
HUNK
ICK
IKK-epsilon
INSR
IRAK1
IRAK3
IRAK4
JAK1(JH2domain-pseudokinase)
JAK2(JH1domain-catalytic)
JAK3(JH1domain-catalytic)
LCK
LKB1
LOK
MAK
MAP3K4
MAP4K3
MAP4K4
MAP4K5
MEK1
MEK2
MEK5
MERTK
MET
MET
MINK
MST1R
MST2
MYLK2
NEK2
PAK1
PAK3
PAK7
PCTK1
PCTK2
PCTK3
PDGFRA
PDGFRB
PFTAIRE2
PFTK1
PHKG1
PHKG2
PIP5K1A
PIP5K2B
PLK4
PRP4
PYK2
RET
RET
RIOK1
RIOK3
RIPK1
RPS6KA5(Kin.Dom.2-C-terminal)
SIK2
SLK
SNARK
SRPK1
SRPK2
SRPK3
STK33
TAOK1
TAOK2
TAOK3
TBK1
TIE1
TNIK
TRKA
TRKB
TRKC
TSSK1B
TYRO3
ULK1
ULK2
YES
YSK4
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